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Main.PHARMA..Drug BioAvailability.Oral Drug BioAvailability.Improvement..Essential Oils (USA.A).Patent.Literature (Claims Etc.).Claim 1: Oral BioAvailability of.Hydrophobic Drug Increase Method:.Co-Adm. Drug & Essential Oil or.Essential Oil Component to provide.Concn. of Essential Oil or Comp. in.Gut > than Concn. that Reduces.Cyclosporin (C) to Hydroxylated (C.) Conversion by 10% in Assay Contg..Rat Liver Microsomes (250 .mu.g).Cyclosporin (1 .mu.M),.& NADPH (1 mM) in.Sodium Phosphate Buffer (1 ml 0.1M).pH = 7.4. Claim 3: Pharma. Compn.:.Carrier, Drug & Essential Oil..Claim 5: Essential Oil or Component.as Counter-Ion of Drug. Claim 6:.Essential Oil or Component.Covalently Linked to Drug..Patent Assignee |